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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
EPHB6 (
O15197
),
reference kinase: EPHB4
(
P54760
)
Kinase group
TK
Number of conformation types
2
Number of structural templates
10 (
Total 265 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
2
2VX0A_7X7
(EPHB4)
TK
2,4-Pyrimidi...
I
6
70
16
A
2VX0A_7X7
(EPHB4)
TK
2,4-Pyrimidi...
I
6
70
16
6
70
16
A
2VWYA_7X5
(EPHB4)
TK
2,4-Pyrimidi...
I
1
38
0
1
38
0
B
8
2VWUA_7X1
(EPHB4)
TK
Chlorobenzod...
I
77
287
111
B
2VWUA_7X1
(EPHB4)
TK
Chlorobenzod...
I
77
287
111
77
287
111
B
2X9FA_X9F
(EPHB4)
TK
X9F
I
46
19
86
46
19
86
B
2VX1A_7X8
(EPHB4)
TK
DB07256
I
19
37
15
19
37
15
B
2VWVA_7X3
(EPHB4)
TK
2vwv
I
13
60
55
13
60
55
B
2VWWA_7X2
(EPHB4)
TK
2vww
I
12
58
55
12
58
55
B
2XVDA_AS6
(EPHB4)
TK
{4-Methyl-3-...
I
4
26
10
4
26
10
B
2VWXA_7X4
(EPHB4)
TK
2,4-Pyrimidi...
I
1
26
0
1
26
0
B
2VWZA_7X6
(EPHB4)
TK
DB07254
I
1
23
0
1
23
0