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KIDFamMap: Kinase-inhibitor-disease family map
Statistics
6 kinase conformation types
and 1208 kinase-inhibitor families
962 kinase-inhibitor-disease relationships
399 human protein kinases
35,788 kinase inhibitors
186,985 kinase-inhibitor assays
55,603 kinase-inhibitor interactions (<=10uM)
339 diseases
638 disease allelic variants
updated at August 23, 2012
Search by kinase
Disease
Compound
Kinase
Input a kinase name (Ex:
ABL1
)
Input a kinase sequence (sequence in FASTA format
)
>ABL1 GMSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEDTMEVEEFLKE AAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVNAVVLLYMATQ ISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAPAGAKFPIKWT APESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPE KVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELGKQ
Browse by Group:
Group
TK (84)
TKL (27)
AGC (56)
Other (32)
CAMK (46)
CMGC (59)
CK1 (8)
STE (28)
Alphabet:
Alphabet
A (21)
B (8)
C (53)
D (14)
E (17)
F (12)
G (8)
H (5)
I (8)
J (3)
K (6)
L (6)
M (46)
N (16)
O (2)
P (52)
R (15)
S (27)
T (13)
U (2)
V (1)
W (2)
Y (1)
Z (2)
All protein kinases
AURKA
AURKB
AURKC
BUB1
CAMKK1
CAMKK2
EIF2AK2
ERN1
ERN2
GSG2
NEK1
NEK10
NEK11
NEK2
NEK3
NEK4
NEK5
NEK6
NEK7
NEK8
NEK9
PLK1
PLK2
PLK3
PLK4
STK16
STK36
TTK
ULK2
ULK3
WEE1
WEE2
ACVR1
ACVR1B
ACVR1C
ACVR2A
ACVRL1
AMHR2
ARAF
BMPR1A
BMPR1B
BMPR2
BRAF
ILK
IRAK1
IRAK4
KIAA1804
KSR1
KSR2
MAP3K10
MAP3K11
MAP3K12
MAP3K13
MAP3K7
MAP3K9
RAF1
TGFBR1
TGFBR2
ZAK
AATK
ABL1
ABL2
ALK
AXL
BLK
BMX
BTK
CSF1R
CSK
DDR1
DDR2
EGFR
EPHA1
EPHA10
EPHA2
EPHA3
EPHA7
EPHB1
EPHB2
EPHB3
EPHB4
EPHB6
ERBB2
ERBB3
ERBB4
FER
FES
FGFR1
FGFR2
FGFR3
FGFR4
FGR
FLT1
FLT4
FRK
FYN
HCK
IGF1R
INSR
INSRR
ITK
JAK1
JAK2
JAK3
KDR
KIT
LCK
LMTK3
LTK
LYN
MATK
MERTK
MET
MST1R
MUSK
NTRK1
NTRK2
NTRK3
PDGFRA
PDGFRB
PTK2
PTK2B
PTK6
PTK7
RET
ROR1
ROR2
ROS1
RYK
SRC
SRMS
STYK1
SYK
TEC
TEK
TIE1
TNK1
TNK2
TXK
TYK2
TYRO3
YES1
ZAP70
ALS2CR2
MAP2K1
MAP2K2
MAP2K3
MAP2K4
MAP2K5
MAP2K6
MAP4K3
MAP4K4
MAP4K5
MINK1
MST4
MYO3A
MYO3B
NRK
OXSR1
PAK1
PAK2
PAK3
PAK4
PAK7
SLK
STK10
STK24
STK25
STK39
STRADA
TNIK
CCRK
CDC2
CDC2L5
CDC2L6
CDK10
CDK11A
CDK15
CDK2
CDK3
CDK5
CDK6
CDK7
CDK8
CDK9
CDKL1
CDKL2
CDKL3
CDKL4
CDKL5
CLK1
CLK2
CLK3
CLK4
CRKRS
CSNK2A1
CSNK2A2
DYRK1A
DYRK1B
DYRK2
DYRK3
DYRK4
GSK3A
GSK3B
HIPK1
HIPK2
HIPK3
HIPK4
ICK
MAK
MAPK1
MAPK10
MAPK11
MAPK12
MAPK14
MAPK15
MAPK3
MAPK7
MAPK8
MAPK9
NLK
PCTK1
PCTK2
PCTK3
PFTK1
PRPF4B
RAGE
SRPK1
SRPK2
SRPK3
CSNK1A1
CSNK1A1L
CSNK1D
CSNK1E
CSNK1G1
CSNK1G2
CSNK1G3
VRK1
CAMK1
CAMK1D
CAMK1G
CAMK2A
CAMK2B
CAMK2D
CAMK2G
CAMK4
CAMKV
CASK
CHEK1
CHEK2
DAPK1
DAPK2
DAPK3
DCLK1
DCLK2
DCLK3
KALRN
LOC729871
MAPKAPK2
MAPKAPK3
MELK
MKNK2
MYLK
MYLK2
MYLK3
MYLK4
OBSCN
PASK
PIM1
PIM2
PIM3
PNCK
PRKAA1
PRKAA2
PRKD1
PRKD2
PRKD3
PSKH1
PSKH2
STK11
STK17A
STK17B
STK33
TRIO
ADRBK1
ADRBK2
AKT1
AKT2
AKT3
CDC42BPA
CDC42BPB
CDC42BPG
CIT
DMPK
FLJ25006
GRK1
GRK4
GRK5
GRK6
GRK7
LOC375449
MAST1
MAST2
MAST3
PDPK1
PKN1
PKN2
PKN3
PRKACA
PRKACB
PRKACG
PRKCA
PRKCB
PRKCD
PRKCE
PRKCG
PRKCH
PRKCI
PRKCQ
PRKCZ
PRKG1
PRKG2
PRKX
PRKY
ROCK1
ROCK2
RPS6KA1
RPS6KA2
RPS6KA3
RPS6KA4
RPS6KA5
RPS6KA6
SGK1
SGK2
SGK3
STK32A
STK32B
STK32C
STK38
STK38L
AATK
ABL1
ABL2
ALK
AXL
ACVR1
ACVR1B
ACVR1C
ACVR2A
ACVRL1
AMHR2
ARAF
ADRBK1
ADRBK2
AKT1
AKT2
AKT3
AURKA
AURKB
AURKC
ALS2CR2
BLK
BMX
BTK
BMPR1A
BMPR1B
BMPR2
BRAF
BUB1
CSF1R
CSK
CDC42BPA
CDC42BPB
CDC42BPG
CIT
CAMKK1
CAMKK2
CAMK1
CAMK1D
CAMK1G
CAMK2A
CAMK2B
CAMK2D
CAMK2G
CAMK4
CAMKV
CASK
CHEK1
CHEK2
CCRK
CDC2
CDC2L5
CDC2L6
CDK10
CDK11A
CDK15
CDK2
CDK3
CDK5
CDK6
CDK7
CDK8
CDK9
CDKL1
CDKL2
CDKL3
CDKL4
CDKL5
CLK1
CLK2
CLK3
CLK4
CRKRS
CSNK2A1
CSNK2A2
CSNK1A1
CSNK1A1L
CSNK1D
CSNK1E
CSNK1G1
CSNK1G2
CSNK1G3
DDR1
DDR2
DMPK
DAPK1
DAPK2
DAPK3
DCLK1
DCLK2
DCLK3
DYRK1A
DYRK1B
DYRK2
DYRK3
DYRK4
EGFR
EPHA1
EPHA10
EPHA2
EPHA3
EPHA7
EPHB1
EPHB2
EPHB3
EPHB4
EPHB6
ERBB2
ERBB3
ERBB4
EIF2AK2
ERN1
ERN2
FER
FES
FGFR1
FGFR2
FGFR3
FGFR4
FGR
FLT1
FLT4
FRK
FYN
FLJ25006
GRK1
GRK4
GRK5
GRK6
GRK7
GSG2
GSK3A
GSK3B
HCK
HIPK1
HIPK2
HIPK3
HIPK4
IGF1R
INSR
INSRR
ITK
ILK
IRAK1
IRAK4
ICK
JAK1
JAK2
JAK3
KDR
KIT
KIAA1804
KSR1
KSR2
KALRN
LCK
LMTK3
LTK
LYN
LOC375449
LOC729871
MATK
MERTK
MET
MST1R
MUSK
MAP3K10
MAP3K11
MAP3K12
MAP3K13
MAP3K7
MAP3K9
MAST1
MAST2
MAST3
MAPKAPK2
MAPKAPK3
MELK
MKNK2
MYLK
MYLK2
MYLK3
MYLK4
MAK
MAPK1
MAPK10
MAPK11
MAPK12
MAPK14
MAPK15
MAPK3
MAPK7
MAPK8
MAPK9
MAP2K1
MAP2K2
MAP2K3
MAP2K4
MAP2K5
MAP2K6
MAP4K3
MAP4K4
MAP4K5
MINK1
MST4
MYO3A
MYO3B
NTRK1
NTRK2
NTRK3
NEK1
NEK10
NEK11
NEK2
NEK3
NEK4
NEK5
NEK6
NEK7
NEK8
NEK9
NLK
NRK
OBSCN
OXSR1
PDGFRA
PDGFRB
PTK2
PTK2B
PTK6
PTK7
PDPK1
PKN1
PKN2
PKN3
PRKACA
PRKACB
PRKACG
PRKCA
PRKCB
PRKCD
PRKCE
PRKCG
PRKCH
PRKCI
PRKCQ
PRKCZ
PRKG1
PRKG2
PRKX
PRKY
PLK1
PLK2
PLK3
PLK4
PASK
PIM1
PIM2
PIM3
PNCK
PRKAA1
PRKAA2
PRKD1
PRKD2
PRKD3
PSKH1
PSKH2
PCTK1
PCTK2
PCTK3
PFTK1
PRPF4B
PAK1
PAK2
PAK3
PAK4
PAK7
RET
ROR1
ROR2
ROS1
RYK
RAF1
ROCK1
ROCK2
RPS6KA1
RPS6KA2
RPS6KA3
RPS6KA4
RPS6KA5
RPS6KA6
RAGE
SRC
SRMS
STYK1
SYK
SGK1
SGK2
SGK3
STK32A
STK32B
STK32C
STK38
STK38L
STK16
STK36
STK11
STK17A
STK17B
STK33
SRPK1
SRPK2
SRPK3
SLK
STK10
STK24
STK25
STK39
STRADA
TEC
TEK
TIE1
TNK1
TNK2
TXK
TYK2
TYRO3
TGFBR1
TGFBR2
TTK
TRIO
TNIK
ULK2
ULK3
VRK1
WEE1
WEE2
YES1
ZAP70
ZAK