|
Select Template |
Comformation Type |
No. of Templates |
Representative Template |
Kinase Group |
Representative Inhibitor |
Inhibitor Type |
No. of Kinases |
No. of Inhibitors |
No. of Diseases |
|
A |
178
|
3DOGA_NNN (CDK2) |
CMGC |
NSC743927 |
I |
50 |
239
| 48 |
|
A |
3DOGA_NNN (CDK2) |
CMGC |
NSC743927 |
I |
50 |
239 |
48 |
50 |
239 |
48 |
|
A |
2Z7SA_P01 (RPS6KA1) |
CMGC |
Lopac0_000938 |
I |
32 |
214 |
49 |
32 |
214 |
49 |
|
A |
3GUBA_GUB (DAPK1) |
CMGC |
2,6,9-Trisub... |
I |
17 |
129 |
35 |
17 |
129 |
35 |
|
A |
3LQ5A_SLQ (CDK9) |
CMGC |
Roscovitine |
I |
25 |
130 |
37 |
25 |
130 |
37 |
|
A |
3DDPA_RC8 (CDK2) |
CMGC |
Roscovitine |
I |
42 |
133 |
57 |
42 |
133 |
57 |
|
A |
2BROA_DF2 (CHEK1) |
CMGC |
pyrrolopyrim... |
I |
29 |
109 |
40 |
29 |
109 |
40 |
|
A |
2BRNA_DF1 (CHEK1) |
CMGC |
pyrrolopyrim... |
I |
30 |
119 |
42 |
30 |
119 |
42 |
|
A |
1G5SA_I17 (CDK2) |
CMGC |
H724 |
I |
43 |
170 |
58 |
43 |
170 |
58 |
|
A |
2BRMA_DFZ (CHEK1) |
CMGC |
DFZ |
I |
21 |
88 |
36 |
21 |
88 |
36 |
|
A |
3AC3A_KSH (LCK) |
CMGC |
imidazo[1,2-... |
I |
13 |
105 |
37 |
13 |
105 |
37 |
|
A |
2WIHA_P48 (CDK2) |
CMGC |
VX_680 |
I |
111 |
425 |
105 |
111 |
425 |
105 |
|
A |
1PYEA_PM1 (CDK2) |
CMGC |
AC1NRCTO |
I |
10 |
54 |
35 |
10 |
54 |
35 |
|
A |
2ZM4A_KSM (LCK) |
CMGC |
BMS-279700 |
I |
25 |
179 |
75 |
25 |
179 |
75 |
|
A |
1BL7A_SB4 (MAPK14) |
CMGC |
SB220025 |
I |
22 |
159 |
29 |
22 |
159 |
29 |
|
A |
1OUKA_084 (MAPK14) |
CMGC |
1ouk |
I |
24 |
139 |
46 |
24 |
139 |
46 |
|
A |
1Z57A_DBQ (CLK1) |
CMGC |
Debromohymen... |
I |
9 |
21 |
25 |
9 |
21 |
25 |
|
A |
1ZLTA_HYM (CHEK1) |
CMGC |
10E-Hymenial... |
I |
15 |
31 |
31 |
15 |
31 |
31 |
|
A |
2C3JA_DBQ (CHEK1) |
CMGC |
Debromohymen... |
I |
14 |
33 |
31 |
14 |
33 |
31 |
|
A |
2CN8A_DBQ (CHEK2) |
CMGC |
Debromohymen... |
I |
11 |
33 |
29 |
11 |
33 |
29 |
|
A |
1U4DA_DBQ (TNK2) |
CMGC |
Debromohymen... |
I |
4 |
19 |
13 |
4 |
19 |
13 |
|
A |
2W17A_I19 (CDK2) |
CMGC |
DB07936 |
I |
25 |
134 |
47 |
25 |
134 |
47 |
|
A |
1OI9A_N20 (CDK2) |
CMGC |
NU-6086 |
I |
52 |
80 |
61 |
52 |
80 |
61 |
|
A |
1Q3WA_ATU (GSK3B) |
CMGC |
alsterpaullone |
I |
24 |
28 |
19 |
24 |
28 |
19 |
|
A |
2ZM1A_KSF (LCK) |
CMGC |
DB08055 |
I |
17 |
153 |
56 |
17 |
153 |
56 |
|
A |
3OT3A_22K (CHEK1) |
CMGC |
INCB18424 |
I |
13 |
30 |
13 |
13 |
30 |
13 |
|
A |
2BRGA_DFY (CHEK1) |
CMGC |
DFY |
I |
18 |
33 |
32 |
18 |
33 |
32 |
|
A |
2VV9A_IM9 (CDK2) |
CMGC |
2vv9 |
I |
19 |
61 |
36 |
19 |
61 |
36 |
|
A |
3BLRA_CPB (CDK9) |
CMGC |
BIIVYFLTOXDA... |
I |
48 |
17 |
41 |
48 |
17 |
41 |
|
A |
3BYOA_AM9 (LCK) |
CMGC |
AC1NS8OV |
I |
28 |
144 |
90 |
28 |
144 |
90 |
|
A |
2J51A_DKI (SLK) |
CMGC |
5-AMINO-3-{[... |
I |
90 |
11 |
103 |
90 |
11 |
103 |
|
A |
2JFLA_DKI (SLK) |
CMGC |
5-AMINO-3-{[... |
I |
90 |
11 |
103 |
90 |
11 |
103 |
|
A |
3BHHA_5CP (CAMK2B) |
CMGC |
DCL001071 |
I |
17 |
45 |
22 |
17 |
45 |
22 |
|
A |
3EOCA_T2A (CDK2) |
CMGC |
5-methyl-7-p... |
I |
42 |
148 |
62 |
42 |
148 |
62 |
|
A |
2WU6A_DKI (CLK3) |
CMGC |
5-AMINO-3-{[... |
I |
26 |
9 |
26 |
26 |
9 |
26 |
|
A |
2BRBA_PFQ (CHEK1) |
CMGC |
2-[(5,6-DIPH... |
I |
8 |
32 |
23 |
8 |
32 |
23 |
|
A |
2C5NA_CK8 (CDK2) |
CMGC |
CK8 |
I |
14 |
49 |
26 |
14 |
49 |
26 |
|
A |
3LM0A_EBD (STK17B) |
CMGC |
DCL001071 |
I |
20 |
106 |
24 |
20 |
106 |
24 |
|
A |
2WEVA_CK7 (CDK2) |
CMGC |
CK7 |
I |
8 |
23 |
17 |
8 |
23 |
17 |
|
A |
3MVMA_39P (MAPK14) |
CMGC |
39P |
I |
24 |
247 |
38 |
24 |
247 |
38 |
|
A |
2JEDA_LG8 (PRKCQ) |
CMGC |
5-Arylidene-... |
I |
67 |
19 |
87 |
67 |
19 |
87 |
|
A |
3BHYA_7CP (DAPK3) |
CMGC |
AT_7519 |
I |
4 |
12 |
3 |
4 |
12 |
3 |
|
A |
3AC8A_KSK (LCK) |
CMGC |
Staurosporine |
I |
12 |
96 |
29 |
12 |
96 |
29 |
|
A |
1UV5A_BRW (GSK3B) |
CMGC |
6-bromoindir... |
I |
27 |
37 |
28 |
27 |
37 |
28 |
|
A |
3MVLA_38P (MAPK14) |
CMGC |
38P |
I |
50 |
308 |
44 |
50 |
308 |
44 |
|
A |
2EUFB_LQQ (CDK6) |
CMGC |
Pyrido-[2,3-... |
I |
13 |
122 |
50 |
13 |
122 |
50 |
|
A |
1ZYSA_199 (CHEK1) |
CMGC |
2,4-Diamino-... |
I |
31 |
92 |
52 |
31 |
92 |
52 |
|
A |
3KVWA_IRB (DYRK2) |
CMGC |
CI_1040 |
I |
15 |
36 |
12 |
15 |
36 |
12 |
|
A |
2X81A_ZZL (AURKA) |
CMGC |
MLN8054 |
I |
22 |
24 |
64 |
22 |
24 |
64 |
|
A |
3AC2A_KSE (LCK) |
CMGC |
Staurosporine |
I |
12 |
96 |
29 |
12 |
96 |
29 |
|
A |
1XJDA_STU (PRKCQ) |
CMGC |
staurosporine |
I |
121 |
101 |
106 |
121 |
101 |
106 |
|
A |
3CKXA_STU (STK24) |
CMGC |
staurosporine |
I |
176 |
104 |
141 |
176 |
104 |
141 |
|
A |
2VTQA_LZA (CDK2) |
CMGC |
pyrazole dia... |
I |
36 |
25 |
31 |
36 |
25 |
31 |
|
A |
2UV2A_GVD (SLK) |
CMGC |
pyrido[4,3-d... |
I |
21 |
80 |
62 |
21 |
80 |
62 |
|
A |
1YVJA_4ST (JAK3) |
CMGC |
staurosporine |
I |
96 |
90 |
126 |
96 |
90 |
126 |
|
A |
3FMEA_STU (MAP2K6) |
CMGC |
staurosporine |
I |
28 |
15 |
20 |
28 |
15 |
20 |
|
A |
2VTTA_LZD (CDK2) |
CMGC |
pyrazole dia... |
I |
158 |
42 |
111 |
158 |
42 |
111 |
|
A |
2VN9A_GVD (CAMK2D) |
CMGC |
pyrido[4,3-d... |
I |
16 |
75 |
24 |
16 |
75 |
24 |
|
A |
3GC7A_B45 (MAPK14) |
CMGC |
Sunitinib |
I |
5 |
63 |
16 |
5 |
63 |
16 |
|
A |
3E87A_G95 (AKT2) |
CMGC |
AG_013736 |
I |
9 |
42 |
28 |
9 |
42 |
28 |
|
A |
1Q3DA_STU (GSK3B) |
CMGC |
staurosporine |
I |
115 |
71 |
61 |
115 |
71 |
61 |
|
A |
3HMOA_STU (TTK) |
CMGC |
staurosporine |
I |
27 |
50 |
20 |
27 |
50 |
20 |
|
A |
3GC8A_B45 (MAPK11) |
CMGC |
Sunitinib |
I |
4 |
61 |
14 |
4 |
61 |
14 |
|
A |
1QPDA_STU (LCK) |
CMGC |
staurosporine |
I |
115 |
76 |
126 |
115 |
76 |
126 |
|
A |
2HZ4A_4ST (ABL1) |
CMGC |
staurosporine |
I |
159 |
103 |
156 |
159 |
103 |
156 |
|
A |
3GC9A_B45 (MAPK11) |
CMGC |
Sunitinib |
I |
4 |
61 |
14 |
4 |
61 |
14 |
|
A |
1AQ1A_STU (CDK2) |
CMGC |
staurosporine |
I |
195 |
76 |
118 |
195 |
76 |
118 |
|
A |
1QPJA_STU (LCK) |
CMGC |
staurosporine |
I |
115 |
76 |
126 |
115 |
76 |
126 |
|
A |
3A4OX_STU (LYN) |
CMGC |
staurosporine |
I |
73 |
70 |
88 |
73 |
70 |
88 |
|
A |
1SM2A_STU (ITK) |
CMGC |
staurosporine |
I |
99 |
104 |
128 |
99 |
104 |
128 |
|
A |
1NVRA_STU (CHEK1) |
CMGC |
staurosporine |
I |
179 |
71 |
79 |
179 |
71 |
79 |
|
A |
1SNUA_STU (ITK) |
CMGC |
staurosporine |
I |
99 |
104 |
128 |
99 |
104 |
128 |
|
A |
3EQRA_T74 (TNK2) |
CMGC |
T74 |
I |
34 |
181 |
86 |
34 |
181 |
86 |
|
A |
2VX3A_D15 (DYRK1A) |
CMGC |
pyrazole-3-y... |
I |
5 |
19 |
18 |
5 |
19 |
18 |
|
A |
2WO6A_D15 (DYRK1A) |
CMGC |
pyrazole-3-y... |
I |
5 |
19 |
18 |
5 |
19 |
18 |
|
A |
1PKDA_UCN (CDK2) |
CMGC |
UCN 02 |
I |
195 |
67 |
118 |
195 |
67 |
118 |
|
A |
3E8DA_G98 (AKT2) |
CMGC |
Roscovitine |
I |
5 |
19 |
21 |
5 |
19 |
21 |
|
A |
3EZRA_EZR (CDK2) |
CMGC |
indazole-ben... |
I |
30 |
145 |
62 |
30 |
145 |
62 |
|
A |
3PJ3A_04L (BTK) |
CMGC |
Imatinib |
II |
99 |
113 |
134 |
99 |
113 |
134 |
|
A |
2HY81_1ST (PAK1) |
CMGC |
UCN 02 |
I |
58 |
20 |
75 |
58 |
20 |
75 |
|
A |
2VU3A_LZE (CDK2) |
CMGC |
AT7519 |
I |
35 |
22 |
29 |
35 |
22 |
29 |
|
A |
3AD6A_KSC (LCK) |
CMGC |
Erlotinib |
I |
13 |
120 |
36 |
13 |
120 |
36 |
|
A |
1BMKA_SB5 (MAPK14) |
CMGC |
SB-218655 |
I |
14 |
116 |
34 |
14 |
116 |
34 |
|
A |
3AC1A_KZI (LCK) |
CMGC |
Staurosporine |
I |
11 |
80 |
32 |
11 |
80 |
32 |
|
A |
3EZVA_EZV (CDK2) |
CMGC |
EZV |
I |
36 |
194 |
65 |
36 |
194 |
65 |
|
A |
1NVQA_UCN (CHEK1) |
CMGC |
UCN 02 |
I |
179 |
65 |
79 |
179 |
65 |
79 |
|
A |
3F5XA_EZV (CDK2) |
CMGC |
EZV |
I |
36 |
194 |
65 |
36 |
194 |
65 |
|
A |
1H1QA_2A6 (CDK2) |
CMGC |
NU-6094 |
I |
10 |
50 |
25 |
10 |
50 |
25 |
|
A |
3AC5A_KZM (LCK) |
CMGC |
Erlotinib |
I |
11 |
120 |
27 |
11 |
120 |
27 |
|
A |
2R3NA_SCZ (CDK2) |
CMGC |
AC1LZZHM |
I |
46 |
175 |
57 |
46 |
175 |
57 |
|
A |
1QPEA_PP2 (LCK) |
CMGC |
AG 1879 |
I |
29 |
63 |
51 |
29 |
63 |
51 |
|
A |
3EIDA_PO5 (CDK2) |
CMGC |
AC1O6YZF |
I |
63 |
211 |
77 |
63 |
211 |
77 |
|
A |
2HXLA_422 (CHEK1) |
CMGC |
DB07075 |
I |
15 |
95 |
36 |
15 |
95 |
36 |
|
A |
3GFEA_P37 (MAPK14) |
CMGC |
DB08349 |
I |
11 |
83 |
29 |
11 |
83 |
29 |
|
A |
3D94A_D94 (IGF1R) |
CMGC |
3-[3-(4-Meth... |
II |
7 |
75 |
28 |
7 |
75 |
28 |
|
A |
2WIPA_P49 (CDK2) |
CMGC |
DB08355 |
I |
14 |
101 |
37 |
14 |
101 |
37 |
|
A |
3DT1A_P40 (MAPK14) |
CMGC |
DB08351 |
II |
18 |
69 |
32 |
18 |
69 |
32 |
|
A |
2C5VA_CK4 (CDK2) |
CMGC |
4-(2,4-DIMET... |
I |
10 |
22 |
18 |
10 |
22 |
18 |
|
A |
1YQJA_6NP (MAPK14) |
CMGC |
AMG_706 |
I |
19 |
102 |
43 |
19 |
102 |
43 |
|
A |
2XYNA_VX6 (ABL2) |
CMGC |
VX-680 |
I |
79 |
101 |
105 |
79 |
101 |
105 |
|
A |
2C6TA_DT5 (CDK2) |
CMGC |
2c6m |
I |
8 |
40 |
39 |
8 |
40 |
39 |
|
A |
3E5AA_VX6 (AURKA) |
CMGC |
VX-680 |
I |
57 |
107 |
93 |
57 |
107 |
93 |
|
A |
3NR9A_NR9 (CLK2) |
CMGC |
Cdk1 Inhibit... |
I |
6 |
5 |
19 |
6 |
5 |
19 |
|
A |
3BYMA_AM0 (LCK) |
CMGC |
triazine 34 |
I |
39 |
145 |
100 |
39 |
145 |
100 |
|
A |
3LHJA_LHJ (MAPK14) |
CMGC |
LHJ |
I |
8 |
89 |
18 |
8 |
89 |
18 |
|
A |
2F4JA_VX6 (ABL1) |
CMGC |
VX-680 |
I |
110 |
109 |
134 |
110 |
109 |
134 |
|
A |
3BHVA_VAR (CDK2) |
CMGC |
Meridianin A |
I |
5 |
8 |
16 |
5 |
8 |
16 |
|
A |
2OW3A_BIM (GSK3B) |
CMGC |
LY_333531 |
I |
62 |
139 |
51 |
62 |
139 |
51 |
|
A |
3DS6A_A17 (MAPK14) |
CMGC |
3ds6 |
II |
21 |
146 |
34 |
21 |
146 |
34 |
|
A |
2XM8A_B4W (CHEK2) |
CMGC |
PI_103 |
I |
12 |
54 |
18 |
12 |
54 |
18 |
|
A |
2JAVA_5Z5 (NEK2) |
CMGC |
pyrrollylact... |
I |
25 |
40 |
24 |
25 |
40 |
24 |
|
A |
3HRBA_I39 (MAPK14) |
CMGC |
PTK_787 |
I |
4 |
29 |
17 |
4 |
29 |
17 |
|
A |
3PIXA_027 (BTK) |
CMGC |
7-(4-Methylp... |
I |
15 |
33 |
55 |
15 |
33 |
55 |
|
A |
1VYWA_292 (CDK2) |
CMGC |
PNU-292137 I... |
I |
20 |
91 |
38 |
20 |
91 |
38 |
|
A |
3C4FA_C4F (FGFR1) |
CMGC |
AC1O6YNE |
I |
23 |
45 |
56 |
23 |
45 |
56 |
|
A |
2ZJWA_REF (CSNK2A1) |
CMGC |
ellagic acid |
I |
8 |
11 |
23 |
8 |
11 |
23 |
|
A |
2W05A_FRT (CDK2) |
CMGC |
2w05 |
I |
7 |
51 |
14 |
7 |
51 |
14 |
|
A |
2C3LA_IDZ (CHEK1) |
CMGC |
IDZ |
I |
14 |
36 |
26 |
14 |
36 |
26 |
|
A |
3EQFA_KSA (MAP2K1) |
CMGC |
k-252a |
I |
42 |
51 |
57 |
42 |
51 |
57 |
|
A |
3LM5A_QUE (STK17B) |
CMGC |
quercetin |
I |
8 |
15 |
20 |
8 |
15 |
20 |
|
A |
2I0EA_PDS (PRKCB) |
CMGC |
bisindolylma... |
I |
41 |
141 |
45 |
41 |
141 |
45 |
|
A |
1NVSA_UCM (CHEK1) |
CMGC |
SB218078 |
I |
97 |
6 |
53 |
97 |
6 |
53 |
|
A |
2HOGA_710 (CHEK1) |
CMGC |
3-(Indol-2-y... |
I |
33 |
66 |
51 |
33 |
66 |
51 |
|
A |
2B55A_D31 (CDK2) |
CMGC |
D31 |
I |
27 |
87 |
53 |
27 |
87 |
53 |
|
A |
2XEYA_YVQ (CHEK1) |
CMGC |
3-(Indol-2-y... |
I |
13 |
35 |
26 |
13 |
35 |
26 |
|
A |
2VTNA_LZ7 (CDK2) |
CMGC |
pyrazole ami... |
I |
8 |
48 |
24 |
8 |
48 |
24 |
|
A |
2JAMA_J60 (CAMK1G) |
CMGC |
SU11652 |
I |
50 |
65 |
32 |
50 |
65 |
32 |
|
A |
3AC4A_KZL (LCK) |
CMGC |
imidazo[1,2-... |
I |
7 |
86 |
21 |
7 |
86 |
21 |
|
A |
1Q41A_IXM (GSK3B) |
CMGC |
INDIRUBIN-3'... |
I |
9 |
25 |
10 |
9 |
25 |
10 |
|
A |
3NLBA_5BE (CHEK1) |
CMGC |
38P |
I |
45 |
115 |
49 |
45 |
115 |
49 |
|
A |
2XEZA_XEZ (CHEK1) |
CMGC |
CAS396129_53_6 |
I |
16 |
35 |
37 |
16 |
35 |
37 |
|
A |
2XIKA_J60 (STK25) |
CMGC |
SU11652 |
I |
59 |
49 |
65 |
59 |
49 |
65 |
|
A |
3FKLA_FKL (MAPK14) |
CMGC |
38P |
I |
9 |
65 |
23 |
9 |
65 |
23 |
|
A |
1OGUA_ST8 (CDK2) |
CMGC |
ST8 |
I |
31 |
21 |
34 |
31 |
21 |
34 |
|
A |
2XF0A_4UB (CHEK1) |
CMGC |
AC1LCX0J |
I |
12 |
32 |
26 |
12 |
32 |
26 |
|
A |
2BR1A_PFP (CHEK1) |
CMGC |
PFP |
I |
6 |
11 |
14 |
6 |
11 |
14 |
|
A |
1Y57A_MPZ (SRC) |
CMGC |
MPZ |
I |
42 |
155 |
94 |
42 |
155 |
94 |
|
A |
2BHEA_BRY (CDK2) |
CMGC |
BRY |
I |
51 |
31 |
35 |
51 |
31 |
35 |
|
A |
3GU8A_3GU (DAPK1) |
CMGC |
Vidarabine |
I |
14 |
17 |
24 |
14 |
17 |
24 |
|
A |
3FSKA_RO6 (MAPK14) |
CMGC |
SU_14813 |
I |
5 |
10 |
24 |
5 |
10 |
24 |
|
A |
3SD0A_TSK (GSK3B) |
CMGC |
3-(5-Fluoro-... |
I |
9 |
38 |
17 |
9 |
38 |
17 |
|
A |
2UUEA_MTZ (CDK2) |
CMGC |
Kinome_636 |
I |
10 |
5 |
16 |
10 |
5 |
16 |
|
A |
3ITZA_P66 (MAPK14) |
CMGC |
P66 |
II |
15 |
102 |
25 |
15 |
102 |
25 |
|
A |
3RI1A_3RH (FGFR2) |
CMGC |
6-o-tolylqui... |
I |
29 |
33 |
72 |
29 |
33 |
72 |
|
A |
2C3KA_ABO (CHEK1) |
CMGC |
ABO |
I |
15 |
47 |
31 |
15 |
47 |
31 |
|
A |
2ZYBA_KSL (LCK) |
CMGC |
DB08056 |
I |
36 |
172 |
80 |
36 |
172 |
80 |
|
A |
3BQRA_4RB (DAPK3) |
CMGC |
ZINC00285933 |
I |
6 |
12 |
7 |
6 |
12 |
7 |
|
A |
1H1SA_4SP (CDK2) |
CMGC |
nu6102 |
I |
30 |
33 |
30 |
30 |
33 |
30 |
|
A |
1GIHA_1PU (CDK2) |
CMGC |
1PU |
I |
13 |
60 |
35 |
13 |
60 |
35 |
|
A |
1OIUA_N76 (CDK2) |
CMGC |
N76 |
I |
4 |
25 |
16 |
4 |
25 |
16 |
|
A |
1DI9A_MSQ (MAPK14) |
CMGC |
MSQ |
I |
14 |
29 |
29 |
14 |
29 |
29 |
|
A |
2IW8A_4SP (CDK2) |
CMGC |
nu6102 |
I |
30 |
33 |
30 |
30 |
33 |
30 |
|
A |
3NUPA_3NU (CDK6) |
CMGC |
INCB18424 |
I |
15 |
23 |
30 |
15 |
23 |
30 |
|
A |
3IPHA_G11 (MAPK14) |
CMGC |
HMS3303K05 |
I |
57 |
108 |
55 |
57 |
108 |
55 |
|
A |
3ANRA_HRM (DYRK1A) |
CMGC |
HARMINE |
I |
8 |
13 |
18 |
8 |
13 |
18 |
|
A |
1OIYA_N41 (CDK2) |
CMGC |
N41 |
I |
33 |
49 |
34 |
33 |
49 |
34 |
|
A |
2IW9A_4SP (CDK2) |
CMGC |
nu6102 |
I |
30 |
33 |
30 |
30 |
33 |
30 |
|
A |
3BHTA_MFR (CDK2) |
CMGC |
Meridianin A |
I |
9 |
11 |
26 |
9 |
11 |
26 |
|
A |
2C5OA_CK2 (CDK2) |
CMGC |
CK2 |
I |
7 |
6 |
14 |
7 |
6 |
14 |
|
A |
1FVVA_107 (CDK2) |
CMGC |
GW-8510 |
I |
2 |
2 |
5 |
2 |
2 |
5 |
|
A |
2FGIA_PD1 (FGFR1) |
CMGC |
Pyrido[2,3-d... |
I |
24 |
157 |
70 |
24 |
157 |
70 |
|
A |
3ACJA_KSS (LCK) |
CMGC |
6,7-dimethox... |
I |
13 |
7 |
25 |
13 |
7 |
25 |
|
A |
3F88A_3HT (GSK3B) |
CMGC |
SMR000144908 |
I |
4 |
3 |
9 |
4 |
3 |
9 |
|
A |
3D0EA_G93 (AKT2) |
CMGC |
9-N-ethyl-8-... |
I |
30 |
15 |
45 |
30 |
15 |
45 |
|
A |
2HY0A_306 (CHEK1) |
CMGC |
AMG_706 |
I |
23 |
80 |
49 |
23 |
80 |
49 |
|
A |
3BHUA_MHR (CDK2) |
CMGC |
Benzo[c][2,7... |
I |
11 |
13 |
27 |
11 |
13 |
27 |
|
A |
3JY9A_JZH (JAK2) |
CMGC |
atropisomer 1 |
I |
11 |
13 |
32 |
11 |
13 |
32 |
|
A |
3ACKA_KSR (LCK) |
CMGC |
AC1O6YMO |
I |
23 |
42 |
56 |
23 |
42 |
56 |
|
A |
3H9FA_92M (TTK) |
CMGC |
Mps1-IN-2 |
I |
12 |
7 |
6 |
12 |
7 |
6 |
|
A |
3HDMA_MMG (SGK1) |
CMGC |
DB08191 |
I |
3 |
15 |
6 |
3 |
15 |
6 |
|
A |
3FMJA_FMJ (MAPK14) |
CMGC |
Imidazo[1,2-... |
I |
6 |
5 |
36 |
6 |
5 |
36 |
|
A |
2WELA_K88 (CAMK2D) |
CMGC |
su6656 |
I |
30 |
30 |
15 |
30 |
30 |
15 |
|
A |
3L8XA_N4D (MAPK14) |
CMGC |
3cg2 |
I |
91 |
104 |
65 |
91 |
104 |
65 |
|
A |
3HDNA_GMG (SGK1) |
CMGC |
DB07837 |
I |
3 |
14 |
6 |
3 |
14 |
6 |
|
A |
1R0EA_DFN (GSK3B) |
CMGC |
HMS3401D14 |
I |
17 |
17 |
17 |
17 |
17 |
17 |
|
A |
2HZIA_JIN (ABL1) |
CMGC |
PD180970 |
I |
90 |
77 |
120 |
90 |
77 |
120 |
|
A |
3RHXA_3RH (FGFR1) |
CMGC |
6-o-tolylqui... |
I |
27 |
31 |
67 |
27 |
31 |
67 |
|
A |
3E92A_G6A (MAPK14) |
CMGC |
3e92 |
I |
56 |
59 |
55 |
56 |
59 |
55 |
|
A |
3PA3A_C70 (CHEK1) |
CMGC |
2-(4-Chlorop... |
I |
11 |
72 |
16 |
11 |
72 |
16 |
|
|
B |
137
|
1UNLA_RRC (CDK5) |
CMGC |
roscovitine |
I |
45 |
237
| 47 |
|
|