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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
CDC2L5 (
Q14004
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
33 (
Total 13 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
21
2DQ7X_STU
(FYN)
CMGC
staurosporine
I
91
74
124
A
2DQ7X_STU
(FYN)
CMGC
staurosporine
I
91
74
124
91
74
124
A
2VTQA_LZA
(CDK2)
CMGC
pyrazole dia...
I
36
25
31
36
25
31
A
2HY81_1ST
(PAK1)
CMGC
UCN 02
I
58
20
75
58
20
75
A
2VTTA_LZD
(CDK2)
CMGC
pyrazole dia...
I
158
42
111
158
42
111
A
3BLRA_CPB
(CDK9)
CMGC
BIIVYFLTOXDA...
I
48
17
41
48
17
41
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
2HZ4A_4ST
(ABL1)
CMGC
staurosporine
I
159
103
156
159
103
156
A
2VU3A_LZE
(CDK2)
CMGC
AT7519
I
35
22
29
35
22
29
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
3A4OX_STU
(LYN)
CMGC
staurosporine
I
73
70
88
73
70
88
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
1QPDA_STU
(LCK)
CMGC
staurosporine
I
115
76
126
115
76
126
A
2JDRA_L20
(AKT2)
CMGC
A-443654
I
44
255
61
44
255
61
A
1BYGA_STU
(CSK)
CMGC
staurosporine
I
85
72
123
85
72
123
A
1QPJA_STU
(LCK)
CMGC
staurosporine
I
115
76
126
115
76
126
A
1NVQA_UCN
(CHEK1)
CMGC
UCN 02
I
179
65
79
179
65
79
A
1XJDA_STU
(PRKCQ)
CMGC
staurosporine
I
121
101
106
121
101
106
A
3CKXA_STU
(STK24)
CMGC
staurosporine
I
176
104
141
176
104
141
A
2OFUA_1N9
(LCK)
CMGC
2-aminopyrim...
I
55
215
101
55
215
101
A
1NVRA_STU
(CHEK1)
CMGC
staurosporine
I
179
71
79
179
71
79
A
1YVJA_4ST
(JAK3)
CMGC
staurosporine
I
96
90
126
96
90
126
B
12
3D7TA_STU
(CSK)
CMGC
staurosporine
I
70
68
99
B
3D7TA_STU
(CSK)
CMGC
staurosporine
I
70
68
99
70
68
99
B
3EFWA_AK8
(AURKA)
CMGC
3efw
I
100
59
105
100
59
105
B
2VTSA_LZC
(CDK2)
CMGC
DB08140
I
28
54
26
28
54
26
B
1OKYA_STU
(PDPK1)
CMGC
staurosporine
I
179
67
109
179
67
109
B
3NYNA_SGV
(GRK6)
CMGC
SMR000127424
I
54
7
47
54
7
47
B
1OKZA_UCN
(PDPK1)
CMGC
UCN 02
I
179
60
109
179
60
109
B
2FVDA_LIA
(CDK2)
CMGC
[4-Amino-2-[...
I
39
16
29
39
16
29
B
2C6EA_HPM
(AURKA)
CMGC
HPM
I
44
237
90
44
237
90
B
3BKBA_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
3CBLA_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
3CD3A_STU
(FES)
CMGC
staurosporine
I
131
107
138
131
107
138
B
3L9MA_L9M
(PRKACA)
CMGC
VX_680
I
37
65
42
37
65
42