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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
CLK4 (
Q9HAZ1
)
Kinase group
CMGC
Number of conformation types
0
Number of structural templates
52 (
Total 162 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
28
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
A
1AQ1A_STU
(CDK2)
CMGC
staurosporine
I
195
76
118
195
76
118
A
1PKDA_UCN
(CDK2)
CMGC
UCN 02
I
195
67
118
195
67
118
A
1Q3DA_STU
(GSK3B)
CMGC
staurosporine
I
115
71
61
115
71
61
A
2OW3A_BIM
(GSK3B)
CMGC
LY_333531
I
62
139
51
62
139
51
A
2VTTA_LZD
(CDK2)
CMGC
pyrazole dia...
I
158
42
111
158
42
111
A
2WU6A_DKI
(CLK3)
CMGC
5-AMINO-3-{[...
I
26
9
26
26
9
26
A
2R3NA_SCZ
(CDK2)
CMGC
AC1LZZHM
I
46
175
57
46
175
57
A
1R78A_FMD
(CDK2)
CMGC
4-alkynyl ox...
I
127
24
97
127
24
97
A
3DOGA_NNN
(CDK2)
CMGC
NSC743927
I
50
239
48
50
239
48
A
3EOCA_T2A
(CDK2)
CMGC
5-methyl-7-p...
I
42
148
62
42
148
62
A
3ANQA_EHB
(DYRK1A)
CMGC
TG003
I
7
3
2
7
3
2
A
1OGUA_ST8
(CDK2)
CMGC
ST8
I
31
21
34
31
21
34
A
3EIDA_PO5
(CDK2)
CMGC
AC1O6YZF
I
63
211
77
63
211
77
A
1R0EA_DFN
(GSK3B)
CMGC
HMS3401D14
I
17
17
17
17
17
17
A
2VTQA_LZA
(CDK2)
CMGC
pyrazole dia...
I
36
25
31
36
25
31
A
1OIYA_N41
(CDK2)
CMGC
N41
I
33
49
34
33
49
34
A
2VU3A_LZE
(CDK2)
CMGC
AT7519
I
35
22
29
35
22
29
A
1PYEA_PM1
(CDK2)
CMGC
AC1NRCTO
I
10
54
35
10
54
35
A
3DDPA_RC8
(CDK2)
CMGC
Roscovitine
I
42
133
57
42
133
57
A
1G5SA_I17
(CDK2)
CMGC
H724
I
43
170
58
43
170
58
A
2IW6A_QQ2
(CDK2)
CMGC
2iw6
I
112
209
86
112
209
86
A
2IW8A_4SP
(CDK2)
CMGC
nu6102
I
30
33
30
30
33
30
A
3GUBA_GUB
(DAPK1)
CMGC
2,6,9-Trisub...
I
17
129
35
17
129
35
A
2IW9A_4SP
(CDK2)
CMGC
nu6102
I
30
33
30
30
33
30
A
3LQ5A_SLQ
(CDK9)
CMGC
Roscovitine
I
25
130
37
25
130
37
A
3EJ1A_5BP
(CDK2)
CMGC
AC1OCFRV
I
46
92
62
46
92
62
A
2WELA_K88
(CAMK2D)
CMGC
su6656
I
30
30
15
30
30
15
A
1H1SA_4SP
(CDK2)
CMGC
nu6102
I
30
33
30
30
33
30
B
24
2F2CB_AP9
(CDK6)
CMGC
MLS000911551
I
24
147
39
B
2F2CB_AP9
(CDK6)
CMGC
MLS000911551
I
24
147
39
24
147
39
B
2R3OA_2SC
(CDK2)
CMGC
4-(Benzylami...
I
18
36
43
18
36
43
B
3PJ8A_404
(CDK2)
CMGC
imidazo[2,1-...
I
47
223
49
47
223
49
B
2A4LA_RRC
(CDK2)
CMGC
roscovitine
I
50
240
50
50
240
50
B
3DDQA_RRC
(CDK2)
CMGC
roscovitine
I
50
240
50
50
240
50
B
1CKPA_PVB
(CDK2)
CMGC
Purvalanol B
I
35
76
36
35
76
36
B
1UNLA_RRC
(CDK5)
CMGC
roscovitine
I
45
237
47
45
237
47
B
1W0XC_OLO
(CDK2)
CMGC
olomoucine
I
43
195
47
43
195
47
B
3NS9A_NS9
(CDK2)
CMGC
pyrazolo[1,5...
I
44
196
47
44
196
47
B
2A0CX_CK9
(CDK2)
CMGC
purine deriv...
I
45
226
50
45
226
50
B
2R3GA_SC9
(CDK2)
CMGC
2r3j
I
30
137
50
30
137
50
B
2FVDA_LIA
(CDK2)
CMGC
[4-Amino-2-[...
I
39
16
29
39
16
29
B
2C68A_CT6
(CDK2)
CMGC
2c68
I
23
73
43
23
73
43
B
2C6IA_DT1
(CDK2)
CMGC
2c6i
I
27
41
48
27
41
48
B
1H07A_MFP
(CDK2)
CMGC
AC1NAKJQ
I
90
241
80
90
241
80
B
2C69A_CT8
(CDK2)
CMGC
CT8
I
22
62
38
22
62
38
B
2C6OA_4SP
(CDK2)
CMGC
nu6102
I
23
33
27
23
33
27
B
1PMNA_984
(MAPK10)
CMGC
1pmn
I
10
124
20
10
124
20
B
2R3JA_SCJ
(CDK2)
CMGC
2r3j
I
27
99
49
27
99
49
B
1PMQA_880
(MAPK10)
CMGC
1pmq
I
12
105
20
12
105
20
B
2R3KA_SCQ
(CDK2)
CMGC
2r3j
I
28
95
49
28
95
49
B
2R3LA_SCW
(CDK2)
CMGC
2r3j
I
19
63
41
19
63
41
B
1OIRA_HDY
(CDK2)
CMGC
AC1O6YZF
I
51
203
64
51
203
64
B
2R3QA_5SC
(CDK2)
CMGC
2r3j
I
5
13
18
5
13
18