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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
MAP3K11 (
Q16584
)
Kinase group
TKL
Number of conformation types
0
Number of structural templates
27 (
Total 105 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
27
3EQFA_KSA
(MAP2K1)
TKL
k-252a
I
42
51
57
A
3EQFA_KSA
(MAP2K1)
TKL
k-252a
I
42
51
57
42
51
57
A
1AQ1A_STU
(CDK2)
TKL
staurosporine
I
195
76
118
195
76
118
A
1SM2A_STU
(ITK)
TKL
staurosporine
I
99
104
128
99
104
128
A
1SNUA_STU
(ITK)
TKL
staurosporine
I
99
104
128
99
104
128
A
3CKXA_STU
(STK24)
TKL
staurosporine
I
176
104
141
176
104
141
A
1PKDA_UCN
(CDK2)
TKL
UCN 02
I
195
67
118
195
67
118
A
2XIKA_J60
(STK25)
TKL
SU11652
I
59
49
65
59
49
65
A
2VTTA_LZD
(CDK2)
TKL
pyrazole dia...
I
158
42
111
158
42
111
A
3DTCA_VIN
(MAP3K9)
TKL
CEP-6331
I
6
21
16
6
21
16
A
2WIHA_P48
(CDK2)
TKL
VX_680
I
111
425
105
111
425
105
A
1R78A_FMD
(CDK2)
TKL
4-alkynyl ox...
I
127
24
97
127
24
97
A
3DOGA_NNN
(CDK2)
TKL
NSC743927
I
50
239
48
50
239
48
A
2IW6A_QQ2
(CDK2)
TKL
2iw6
I
112
209
86
112
209
86
A
2X2MA_X2M
(RET)
TKL
Semaxanib
I
24
81
59
24
81
59
A
2Z7SA_P01
(RPS6KA1)
TKL
Lopac0_000938
I
32
214
49
32
214
49
A
2IW9A_4SP
(CDK2)
TKL
nu6102
I
30
33
30
30
33
30
A
1VYWA_292
(CDK2)
TKL
PNU-292137 I...
I
20
91
38
20
91
38
A
2BHEA_BRY
(CDK2)
TKL
BRY
I
51
31
35
51
31
35
A
2R3NA_SCZ
(CDK2)
TKL
AC1LZZHM
I
46
175
57
46
175
57
A
2IVUA_ZD6
(RET)
TKL
Vandetanib
I
83
291
121
83
291
121
A
3EJ1A_5BP
(CDK2)
TKL
AC1OCFRV
I
46
92
62
46
92
62
A
2X2KA_X2K
(RET)
TKL
Semaxanib
I
23
30
58
23
30
58
A
1H1SA_4SP
(CDK2)
TKL
nu6102
I
30
33
30
30
33
30
A
1OGUA_ST8
(CDK2)
TKL
ST8
I
31
21
34
31
21
34
A
1OIYA_N41
(CDK2)
TKL
N41
I
33
49
34
33
49
34
A
3DDPA_RC8
(CDK2)
TKL
Roscovitine
I
42
133
57
42
133
57
A
2IW8A_4SP
(CDK2)
TKL
nu6102
I
30
33
30
30
33
30