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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
STK39 (
Q9UEW8
)
Kinase group
STE
Number of conformation types
0
Number of structural templates
27 (
Total 15 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
9
1SM2A_STU
(ITK)
STE
staurosporine
I
99
104
128
A
1SM2A_STU
(ITK)
STE
staurosporine
I
99
104
128
99
104
128
A
1SNUA_STU
(ITK)
STE
staurosporine
I
99
104
128
99
104
128
A
2DQ7X_STU
(FYN)
STE
staurosporine
I
91
74
124
91
74
124
A
2HZ4A_4ST
(ABL1)
STE
staurosporine
I
159
103
156
159
103
156
A
1QPDA_STU
(LCK)
STE
staurosporine
I
115
76
126
115
76
126
A
1QPJA_STU
(LCK)
STE
staurosporine
I
115
76
126
115
76
126
A
3L8XA_N4D
(MAPK14)
STE
3cg2
I
91
104
65
91
104
65
A
3PJ3A_04L
(BTK)
STE
Imatinib
II
99
113
134
99
113
134
A
2H8HA_H8H
(SRC)
STE
Saracatinib
I
91
255
126
91
255
126
B
18
2PE2A_464
(PDPK1)
STE
Indolinone b...
I
134
156
104
B
2PE2A_464
(PDPK1)
STE
Indolinone b...
I
134
156
104
134
156
104
B
3MIYA_B49
(ITK)
STE
Sunitinib
I
70
74
110
70
74
110
B
3CBLA_STU
(FES)
STE
staurosporine
I
131
107
138
131
107
138
B
3CD3A_STU
(FES)
STE
staurosporine
I
131
107
138
131
107
138
B
1OKYA_STU
(PDPK1)
STE
staurosporine
I
179
67
109
179
67
109
B
2ITQA_STU
(EGFR)
STE
staurosporine
I
80
85
106
80
85
106
B
1OKZA_UCN
(PDPK1)
STE
UCN 02
I
179
60
109
179
60
109
B
2ITUA_STU
(EGFR)
STE
staurosporine
I
80
85
106
80
85
106
B
2ITWA_STU
(EGFR)
STE
staurosporine
I
80
85
106
80
85
106
B
3BKBA_STU
(FES)
STE
staurosporine
I
131
107
138
131
107
138
B
2ITZA_IRE
(EGFR)
STE
Gefitinib
I
69
313
99
69
313
99
B
2VWUA_7X1
(EPHB4)
STE
Chlorobenzod...
I
77
287
111
77
287
111
B
3EFWA_AK8
(AURKA)
STE
3efw
I
100
59
105
100
59
105
B
3F5PA_741
(IGF1R)
STE
3-cyanoquino...
I
60
123
81
60
123
81
B
2BMCA_MPY
(AURKA)
STE
PHA-680632
I
107
108
107
107
108
107
B
1H07A_MFP
(CDK2)
STE
AC1NAKJQ
I
90
241
80
90
241
80
B
2ITOA_IRE
(EGFR)
STE
Gefitinib
I
69
313
99
69
313
99
B
2ITYA_IRE
(EGFR)
STE
Gefitinib
I
69
313
99
69
313
99