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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Summary of query kinase
Query kinase
TXK (
P42681
)
Kinase group
TK
Number of conformation types
0
Number of structural templates
77 (
Total 71 inhibitors
)
Select
Template
Comformation
Type
No. of
Templates
Representative
Template
Kinase
Group
Representative
Inhibitor
Inhibitor
Type
No. of
Kinases
No. of
Inhibitors
No. of
Diseases
A
41
2IVUA_ZD6
(RET)
TK
Vandetanib
I
83
291
121
A
2IVUA_ZD6
(RET)
TK
Vandetanib
I
83
291
121
83
291
121
A
2H8HA_H8H
(SRC)
TK
Saracatinib
I
91
255
126
91
255
126
A
2GQGA_1N1
(ABL1)
TK
Dasatinib
I
74
32
117
74
32
117
A
1YVJA_4ST
(JAK3)
TK
staurosporine
I
96
90
126
96
90
126
A
3K54A_1N1
(BTK)
TK
Dasatinib
I
56
32
103
56
32
103
A
1QPDA_STU
(LCK)
TK
staurosporine
I
115
76
126
115
76
126
A
2DQ7X_STU
(FYN)
TK
staurosporine
I
91
74
124
91
74
124
A
3CKXA_STU
(STK24)
TK
staurosporine
I
176
104
141
176
104
141
A
3OCTA_1N1
(BTK)
TK
Dasatinib
I
56
32
103
56
32
103
A
1QPJA_STU
(LCK)
TK
staurosporine
I
115
76
126
115
76
126
A
1SM2A_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
2HZ4A_4ST
(ABL1)
TK
staurosporine
I
159
103
156
159
103
156
A
1SNUA_STU
(ITK)
TK
staurosporine
I
99
104
128
99
104
128
A
1U59A_STU
(ZAP70)
TK
staurosporine
I
96
80
114
96
80
114
A
1XBCA_STU
(SYK)
TK
staurosporine
I
71
72
105
71
72
105
A
1XJDA_STU
(PRKCQ)
TK
staurosporine
I
121
101
106
121
101
106
A
2HY81_1ST
(PAK1)
TK
UCN 02
I
58
20
75
58
20
75
A
2F4JA_VX6
(ABL1)
TK
VX-680
I
110
109
134
110
109
134
A
2XYNA_VX6
(ABL2)
TK
VX-680
I
79
101
105
79
101
105
A
3PJ3A_04L
(BTK)
TK
Imatinib
II
99
113
134
99
113
134
A
1PMEA_SB2
(MAPK1)
TK
SB 203580
I
16
31
26
16
31
26
A
2JIUA_AEE
(EGFR)
TK
GNF-Pf-5343
I
26
170
77
26
170
77
A
2JEDA_LG8
(PRKCQ)
TK
5-Arylidene-...
I
67
19
87
67
19
87
A
2Z7SA_P01
(RPS6KA1)
TK
Lopac0_000938
I
32
214
49
32
214
49
A
3FQSA_585
(SYK)
TK
R-406
I
64
28
102
64
28
102
A
1QCFA_PP1
(HCK)
TK
PP1
I
31
65
68
31
65
68
A
3IKAA_0UN
(EGFR)
TK
2jkk
I
76
120
108
76
120
108
A
2XM8A_B4W
(CHEK2)
TK
PI_103
I
12
54
18
12
54
18
A
1QPEA_PP2
(LCK)
TK
AG 1879
I
29
63
51
29
63
51
A
1M17A_AQ4
(EGFR)
TK
Erlotinib
I
43
166
82
43
166
82
A
3PIYA_585
(BTK)
TK
R-406
I
93
17
123
93
17
123
A
1WZYA_F29
(MAPK1)
TK
AC1O4W7N
I
27
48
33
27
48
33
A
3GENA_B43
(BTK)
TK
7-Cyclopenty...
I
29
110
67
29
110
67
A
2IVVA_PP1
(RET)
TK
PP1
I
27
46
63
27
46
63
A
1OPLA_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
3RI1A_3RH
(FGFR2)
TK
6-o-tolylqui...
I
29
33
72
29
33
72
A
2FO0A_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
2ITTA_AEE
(EGFR)
TK
GNF-Pf-5343
I
26
170
77
26
170
77
A
2ZYBA_KSL
(LCK)
TK
DB08056
I
36
172
80
36
172
80
A
2G2HA_P16
(ABL1)
TK
PD166326
I
89
70
123
89
70
123
A
2HZIA_JIN
(ABL1)
TK
PD180970
I
90
77
120
90
77
120
B
35
2ITOA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
B
2ITOA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2ITYA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2ITZA_IRE
(EGFR)
TK
Gefitinib
I
69
313
99
69
313
99
B
2VWUA_7X1
(EPHB4)
TK
Chlorobenzod...
I
77
287
111
77
287
111
B
3CBLA_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
3CD3A_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
3D7TA_STU
(CSK)
TK
staurosporine
I
70
68
99
70
68
99
B
3LCSA_STU
(ALK)
TK
staurosporine
I
73
100
109
73
100
109
B
2ITQA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
2ITUA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
2ITWA_STU
(EGFR)
TK
staurosporine
I
80
85
106
80
85
106
B
3BKBA_STU
(FES)
TK
staurosporine
I
131
107
138
131
107
138
B
1OKYA_STU
(PDPK1)
TK
staurosporine
I
179
67
109
179
67
109
B
1OKZA_UCN
(PDPK1)
TK
UCN 02
I
179
60
109
179
60
109
B
2X9FA_X9F
(EPHB4)
TK
X9F
I
46
19
86
46
19
86
B
3F5PA_741
(IGF1R)
TK
3-cyanoquino...
I
60
123
81
60
123
81
B
3LW0A_CCX
(IGF1R)
TK
5-vinyl-3-py...
III
53
30
101
53
30
101
B
3P9JA_P9J
(AURKA)
TK
4-[(5-Methyl...
I
32
50
54
32
50
54
B
2XRUA_400
(AURKA)
TK
VX_680
I
33
152
63
33
152
63
B
2PE2A_464
(PDPK1)
TK
Indolinone b...
I
134
156
104
134
156
104
B
2J5FA_DJK
(EGFR)
TK
4-anilinoqui...
I
16
212
45
16
212
45
B
2XM9A_LWH
(CHEK2)
TK
4-(1h-Pyrazo...
I
5
34
17
5
34
17
B
3COHA_83H
(AURKA)
TK
AKI-001
I
79
88
65
79
88
65
B
3H9OA_9BD
(PDPK1)
TK
Benzo[c][2,7...
I
45
68
71
45
68
71
B
2XB7A_GUI
(ALK)
TK
NVP-TAE684
I
71
66
107
71
66
107
B
3EKNA_GS3
(INSR)
TK
pyrrolo[2,3-...
I
90
215
127
90
215
127
B
2ITPA_AEE
(EGFR)
TK
GNF-Pf-5343
I
24
168
73
24
168
73
B
1UNLA_RRC
(CDK5)
TK
roscovitine
I
45
237
47
45
237
47
B
2VX1A_7X8
(EPHB4)
TK
DB07256
I
19
37
15
19
37
15
B
1YOMA_P01
(SRC)
TK
Lopac0_000938
I
27
95
57
27
95
57
B
2WTCA_VGM
(CHEK2)
TK
VGM
I
10
39
19
10
39
19
B
2J6MA_AEE
(EGFR)
TK
GNF-Pf-5343
I
24
168
73
24
168
73
B
2BMCA_MPY
(AURKA)
TK
PHA-680632
I
107
108
107
107
108
107
B
2F57B_23D
(PAK7)
TK
CGP74514A
I
11
77
24
11
77
24
B
3NRMA_NRM
(AURKA)
TK
CAS404828_08_6
I
32
33
60
32
33
60
E
1
3C7QA_XIN
(KDR)
TK
BIBF1120
I
25
56
50
E
3C7QA_XIN
(KDR)
TK
BIBF1120
I
25
56
50
25
56
50