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Diseases
Inhibitor-Anchor Map
Family Anchors
Kinase-Inhibitor Family
Template
Protein
Surface
Ribbon
Inhibitor
MQY
ATP Location
Pocket
ATP
NLP
HAP
CLP
SP
Selected template
Kinase
IGF1R (PDB code: 3O23)
[PDB]
[PDBsum]
Inhibitor
(5s)-5-Methyl-1-(Quinolin-4-Ylmethyl)-3-{4-[(Trifluoromethyl)sulfonyl]phenyl}imidazolidine-2,4-Dione (HET code: MQY)
[PDB]
Summary of KIF 3O23A_MQY
(IGF1R, PDB code:
3O23
, chain A)
Number of family interactions
9
Number of family kinase
2 (
sequence conservation
) (
profiling results
)
Number of family inhibitors
8 (8 are IGF1R inhibitors)
Involved diseases
9 (
show
)
Number of family anchors
All kinase-inhibitor interactions in this family
IGF1R and 8 inhibitors